SCHEMBL13257568

SCHEMBL13257568

N#Cc1c(-c2ccnc(N)c2)sc(-c2nnc(Br)[nH]2)c1-c1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
ROCK1 Q13464 1/20 0.38
DYRK1A Q13627 4/20 0.37
GSK3B P49841 2/20 0.37
GSK3A P49840 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
MET P08581 1/20 0.36
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.33
KDM4E B2RXH2 3/20 0.33
SCN9A Q15858 4/20 0.33
MGAM O43451 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SI P14410 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL954282 0.84 PIK3CA (0.40) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL13105876 0.84 PIK3CA (0.41) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL955529 0.83 TGFBR1 (0.40) PIK3CAMTORGSK3BGSK3AGAA
SCHEMBL955202 0.81 PIK3CA (0.42) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL957625 0.80 IDO1 (0.38) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL952533 0.80 PIK3CA (0.39) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL13256634 0.80 PIK3CA (0.39) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL12947611 0.77 CDC7 (0.44) PIK3CAMTORROCK1DYRK1AGSK3B
SCHEMBL13256970 0.74 PIK3C3 (0.40) PIK3C3SCN9ACYP3A4
SCHEMBL956193 0.73 PIK3CA (0.40) PIK3CAMTORDYRK1AGSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090716-A1 HETEROARYLS AND THEIR USE AS PI3K INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed