SCHEMBL13259386

SCHEMBL13259386

Bc1ccc2c(c1)CN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.72
ESR2 Q92731 6/20 0.72
PKM P14618 1/20 0.51
ABHD6 Q9BV23 4/20 0.48
HDAC6 Q9UBN7 2/20 0.45
HDAC8 Q9BY41 1/20 0.45
NR1H2 P55055 1/20 0.42
NOTUM Q6P988 1/20 0.40
MERTK Q12866 3/20 0.39
AXL P30530 2/20 0.39
TYRO3 Q06418 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4183920 0.84 ESR1 (0.74) ESR1ESR2PKMABHD6MERTK
SCHEMBL29754116 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6
SCHEMBL1641841 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6
SCHEMBL29989790 0.82 ESR1 (0.76) ESR1ESR2PKMABHD6MERTK
SCHEMBL2821470 0.82 ESR1 (0.76) ESR1ESR2PKMABHD6MERTK
SCHEMBL3865684 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6NOTUM
SCHEMBL2616863 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6
SCHEMBL585650 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6
SCHEMBL8266789 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6
SCHEMBL30411956 0.82 ESR1 (0.72) ESR1ESR2PKMABHD6HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093425-A1 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2010-08-19 WO disclosed