SCHEMBL13261024

SCHEMBL13261024

CNC1CCN(C(=O)[C@H](Cc2ccc(C)cc2)NC(=O)C2(c3ccc(O)cc3)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 8/20 0.46
CYP3A4 P08684 6/20 0.45
UGCG Q16739 6/20 0.45
ITGB3 P05106 3/20 0.43
ITGA2B P08514 3/20 0.43
KCNH2 Q12809 1/20 0.43
CYP51A1 Q16850 1/20 0.41
OXTR P30559 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21326358 0.79 CYP3A4 (0.57) AVPR1ACYP3A4UGCGKCNH2OXTR
SCHEMBL21326301 0.79 CYP3A4 (0.57) AVPR1ACYP3A4UGCG
SCHEMBL21326305 0.79 CYP3A4 (0.57) AVPR1ACYP3A4UGCG
SCHEMBL21326359 0.79 CYP3A4 (0.57) AVPR1ACYP3A4UGCGKCNH2OXTR
SCHEMBL21326340 0.76 CYP3A4 (0.54) AVPR1ACYP3A4UGCGOXTR
SCHEMBL21326343 0.76 CYP3A4 (0.54) AVPR1ACYP3A4UGCGOXTR
SCHEMBL13655788 0.74 SMYD3 (0.44) ITGB3ITGA2BCYP51A1
SCHEMBL21326270 0.74 CYP3A4 (0.65) AVPR1ACYP3A4UGCGKCNH2OXTR
SCHEMBL21326274 0.74 CYP3A4 (0.65) AVPR1ACYP3A4UGCGKCNH2OXTR
SCHEMBL21326369 0.74 CYP3A4 (0.65) AVPR1ACYP3A4UGCGKCNH2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091164-A1 INHIBITORS OF GLUCOSYLCERAMIDE SYNTHASE EXELIXIS, INC. (US) 2010-08-12 WO disclosed