SCHEMBL13655788

SCHEMBL13655788

CNC1CCN(C(=O)[C@H](O)Cc2ccc(O)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 7/20 0.44
OPRD1 P41143 1/20 0.43
DPP4 P27487 2/20 0.41
EPHX2 P34913 1/20 0.41
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
CYP51A1 Q16850 1/20 0.39
HDAC8 Q9BY41 2/20 0.39
HPGD P15428 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364597 0.80 SMN1; SMN2 (0.47) OPRD1DPP4ITGB3ITGA2BHDAC8
SCHEMBL5364603 0.80 TPSAB1 (0.44) SMYD3OPRD1DPP4ITGB3ITGA2B
SCHEMBL16002877 0.78 ALDH1A1 (0.52) EPHX2HPGDSIGMAR1
SCHEMBL17207616 0.75 EPHX2 (0.47) DPP4EPHX2
SCHEMBL3145714 0.74 DPP4 (0.57) SMYD3OPRD1DPP4
SCHEMBL13261024 0.74 AVPR1A (0.46) ITGB3ITGA2BCYP51A1
SCHEMBL13772745 0.74 EPHX2 (0.33) SMYD3EPHX2SIGMAR1
SCHEMBL6164884 0.74 OPRD1 (0.60) SMYD3OPRD1DPP4HDAC8
SCHEMBL16003001 0.73 MGLL (0.55) EPHX2
SCHEMBL3142935 0.73 MEN1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108648-A1 Selected CGRP antagonists, method for their manufacture and use as medicines Boehringer Ingelheim International GmbH (DE) 2009-10-14 EP disclosed