SCHEMBL13285191

SCHEMBL13285191

Cc1c(CC(=O)O)c2cc(F)ccc2n1C(=O)c1ccc(F)cc1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.86
AKR1C2 P52895 9/20 0.86
PTGS2 P35354 4/20 0.65
PTGS1 P23219 3/20 0.65
LMNA P02545 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2D6 P10635 2/20 0.62
CYP2C9 P11712 2/20 0.62
HIF1A Q16665 2/20 0.62
NPSR1 Q6W5P4 2/20 0.62
TSHR P16473 1/20 0.62
NFKB1 P19838 1/20 0.62
PTGDR2 Q9Y5Y4 2/20 0.61
AKR1C4 P17516 2/20 0.61
AKR1C1 Q04828 2/20 0.61
ABCB1 P08183 2/20 0.61
KDM4E B2RXH2 1/20 0.61
MEN1 O00255 1/20 0.61
PTGES O14684 1/20 0.61
ABCC3 O15438 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2615155 0.95 AKR1C3 (0.83) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL2615154 0.95 AKR1C3 (0.83) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL2615156 0.93 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL2615153 0.93 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL2997297 0.91 PTGS2 (0.79) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL13802249 0.89 AKR1C3 (0.74) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL5796934 0.88 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL5447453 0.85 AKR1C3 (0.66) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL11658058 0.85 AKR1C3 (0.66) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL11730189 0.85 AKR1C3 (0.66) AKR1C3AKR1C2PTGS2PTGS1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010081036-A2 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-07-15 WO disclosed