SCHEMBL13285286

SCHEMBL13285286

C=C1Nc2cc(CN3CCN(c4ccc(C(=O)NC5CC5)cn4)CC3)cnc2N2CCCC[C@@H]12

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.50
TNK1 Q13470 2/20 0.50
TNK2 Q07912 1/20 0.50
HPGDS O60760 5/20 0.46
ACKR3 P25106 1/20 0.45
SMO Q99835 1/20 0.42
PRKAB2 O43741 2/20 0.41
PRKAG1 P54619 2/20 0.41
PRKAA2 P54646 2/20 0.41
PRKAA1 Q13131 2/20 0.41
PRKAG3 Q9UGI9 2/20 0.41
PRKAG2 Q9UGJ0 2/20 0.41
PRKAB1 Q9Y478 2/20 0.41
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
DRD3 P35462 1/20 0.40
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708792 0.92 PARP1 (0.52) PARP1TNK1TNK2HPGDSACKR3
SCHEMBL13285127 0.90 PARP1 (0.48) PARP1TNK1TNK2ACKR3
SCHEMBL6128547 0.89 PARP1 (0.53) PARP1TNK1TNK2HPGDSACKR3
SCHEMBL705982 0.89 PARP1 (0.53) PARP1TNK1TNK2HPGDSACKR3
SCHEMBL709447 0.83 PARP1 (0.49) PARP1TNK1TNK2ACKR3
SCHEMBL709766 0.82 PARP1 (0.57) PARP1
SCHEMBL708669 0.81 PARP1 (0.44) PARP1TNK1TNK2ACKR3
SCHEMBL709746 0.81 PARP1 (0.51) PARP1TNK1TNK2ACKR3
SCHEMBL709173 0.81 PARP1 (0.48) PARP1TNK1TNK2ACKR3SMO
SCHEMBL706995 0.81 PARP1 (0.48) PARP1TNK1TNK2ACKR3SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010085570-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-07-29 WO disclosed