SCHEMBL13285290

SCHEMBL13285290

C=C1OB(c2cnc(-c3cccc(Cc4nnc5ccc(Oc6ccccc6)nn45)c3)nc2)OC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MET P08581 11/20 0.38
LRRK2 Q5S007 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12224242 0.89 MET (0.41) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL12245595 0.89 SMN1; SMN2 (0.39) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL14724354 0.83 MET (0.36) LMNASMN1; SMN2NPSR1MET
SCHEMBL12224229 0.81 SMN1; SMN2 (0.48) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL12224243 0.81 MET (0.47) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL12245312 0.79 MET (0.44) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL2458149 0.79 MET (0.44) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL12224218 0.77 SMN1; SMN2 (0.40) LMNATSHRHTTSMN1; SMN2NPSR1
SCHEMBL2529571 0.73 MET (0.46) TSHRMET
SCHEMBL12224262 0.71 MET (0.38) SMN1; SMN2NPSR1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072301-A1 3-(3-PYRIMIDINE-2-YL-BENZYL)-[1,2,4] TRIAZOLO [4,3-B] PYRIDAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2010-07-01 WO disclosed