SCHEMBL13285293

SCHEMBL13285293

COC(=O)Cc1c(-c2ccccc2)noc1C(=O)F

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.46
GABRA5 P31644 8/20 0.44
ALDH1A1 P00352 3/20 0.43
NR1H4 Q96RI1 3/20 0.41
KDM4E B2RXH2 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
PPARD Q03181 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13284947 0.92 PTGS1 (0.48) PTGS1GABRA5ALDH1A1NR1H4KDM4E
SCHEMBL12406914 0.82 PTGS1 (0.59) PTGS1GABRA5ALDH1A1NR1H4KDM4E
SCHEMBL13285213 0.82 PTGS1 (0.49) PTGS1GABRA5ALDH1A1NR1H4KDM4E
SCHEMBL2565750 0.77 PTGS1 (0.68) PTGS1GABRA5ALDH1A1KDM4E
SCHEMBL10127870 0.76 GABRA5 (0.49) GABRA5ALDH1A1KDM4EAPOBEC3G
SCHEMBL13285291 0.76 PTGS1 (0.55) PTGS1ALDH1A1KDM4E
SCHEMBL18472810 0.74 PTGS1 (0.49) PTGS1GABRA5ALDH1A1KDM4EAPOBEC3G
SCHEMBL13285289 0.73 PTGS1 (0.45) PTGS1ALDH1A1KDM4EAPOBEC3G
SCHEMBL13285212 0.71 PTGS1 (0.46) PTGS1ALDH1A1KDM4EAPOBEC3G
SCHEMBL2565963 0.71 PPARA (0.47) PTGS1ALDH1A1NR1H4PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8354398-B2 Substituted isoxazole compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-15 US disclosed
WO-2010085581-A1 SUBSTITUTED OXADIAZOLE DERIVATIVES AS S1P AGONISTS IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2010-07-29 WO disclosed