SCHEMBL13296351

SCHEMBL13296351

CCN1C(=O)C(=O)N(Cc2ccc(OC)cc2)C1=O

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 2/20 0.74
GSK3A P49840 2/20 0.60
GSK3B P49841 2/20 0.60
EP300 Q09472 1/20 0.56
PTPN1 P18031 1/20 0.54
CASP3 P42574 2/20 0.54
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 2/20 0.50
BLM P54132 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAPT P10636 1/20 0.50
APAF1 O14727 1/20 0.49
GAA P10253 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
CHRM5 P08912 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117134 0.78 CMA1 (0.77) CMA1GSK3AGSK3BEP300CASP3
SCHEMBL2643216 0.77 CMA1 (0.70) CMA1GSK3AGSK3BCASP3KDM4E
SCHEMBL8331785 0.77 CMA1 (0.70) CMA1GSK3AGSK3BCASP3KDM4E
SCHEMBL3384174 0.75 GSK3A (1.00) CMA1GSK3AGSK3BCASP3KDM4E
SCHEMBL3295317 0.75 CMA1 (0.56) CMA1GSK3AGSK3BEP300PTPN1
SCHEMBL3296532 0.75 MAPT (0.56) CMA1EP300ALDH1A1MAPT
SCHEMBL30296449 0.75 CASP3 (0.88) CMA1CASP3KDM4EMEN1KMT2A
SCHEMBL45154 0.75 CASP3 (0.88) CMA1CASP3KDM4EMEN1KMT2A
SCHEMBL15773124 0.75 KDM4E (0.75) CMA1GSK3AGSK3BCASP3KDM4E
SCHEMBL27488298 0.74 CMA1 (0.59) CMA1GSK3AGSK3BCASP3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7737283-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2010-06-15 US disclosed
US-20090312349-A1 ANTI-INFLAMMATORY MEDICAMENTS DECIPHERA PHARMACEUTICALS, LLC 2009-12-17 US disclosed
US-7531566-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2009-05-12 US disclosed
US-20090105230-A1 Anti-inflammatory medicaments FLYNN DANIEL L 2009-04-23 US disclosed
US-20090075986-A1 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC 2009-03-19 US disclosed
US-20080187978-A1 Anti-inflammatory medicaments FLYNN DANIEL L 2008-08-07 US disclosed
US-20080132506-A1 Anti-inflammatory medicaments FLYNN DANIEL L 2008-06-05 US disclosed
US-20080064688-A1 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC 2008-03-13 US disclosed
US-7342037-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2008-03-11 US disclosed
US-20070191336-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-08-16 US disclosed
US-7202257-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2007-04-10 US disclosed
US-20070037808-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064688-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CMA1 524/4885GSK3A 938/4885GSK3B 1164/4885
US-20090105230-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CMA1 524/4885GSK3A 938/4885GSK3B 1164/4885
US-20090075986-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CMA1 524/4885GSK3A 938/4885GSK3B 1164/4885
US-20070037808-A1 p38 kinase inhibitors MAPK1, MAP3K8, MAP3K1 CMA1 2666/4885GSK3A 715/4885GSK3B 744/4885
US-20090312349-A1 ANTI-INFLAMMATORY MEDICAMENTS ABL2, ABL1, PTK2 CMA1 1396/4885GSK3A 662/4885GSK3B 730/4885
US-20070191336-A1 p38 kinase inhibitors MAPK1, MAP3K8, MAP3K1 CMA1 2666/4885GSK3A 715/4885GSK3B 744/4885
US-20080132506-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CMA1 524/4885GSK3A 938/4885GSK3B 1164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.