SCHEMBL1330304

SCHEMBL1330304

CCNCC(O)COc1ccccc1C(C)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.62
ABCB1 P08183 9/20 0.60
LMNA P02545 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP3A4 P08684 2/20 0.56
KCNK3 O14649 1/20 0.56
SLC22A1 O15245 1/20 0.56
ABCC9 O60706 1/20 0.56
KCNK2 O95069 1/20 0.56
ABCB11 O95342 1/20 0.56
ADRB2 P07550 1/20 0.56
ADRB1 P08588 1/20 0.56
ADRB3 P13945 1/20 0.56
ADRA2C P18825 1/20 0.56
SLC6A2 P23975 1/20 0.56
HTR2A P28223 1/20 0.56
HTR2C P28335 1/20 0.56
SLC6A4 P31645 1/20 0.56
ADRA1A P35348 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10968562 0.85 POLB (0.59) POLBABCB1LMNACYP1A2CYP2D6
SCHEMBL7372331 0.82 POLB (0.56) POLBABCB1LMNACYP1A2CYP2D6
SCHEMBL7363941 0.81 POLB (0.55) POLBABCB1LMNACYP1A2CYP2D6
SCHEMBL11180904 0.80 ABCB1 (0.66) POLBABCB1LMNASMN1; SMN2TP53
SCHEMBL22639704 0.78 POLB (0.98) POLBABCB1LMNAADRB2ADRB1
SCHEMBL22639942 0.78 POLB (0.98) POLBABCB1LMNAADRB2ADRB1
SCHEMBL16727483 0.77 ABCB1 (0.75) POLBABCB1LMNAADRB2ADRB1
SCHEMBL8781936 0.76 NR2E1 (0.71) ABCB1LMNACYP1A2CYP2D6SLC22A1
SCHEMBL3339926 0.76 ABCB1 (0.64) POLBABCB1LMNASMN1; SMN2TP53
SCHEMBL10876890 0.76 ABCB1 (0.57) ABCB1LMNACYP1A2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8323911-B2 High throughput assay for discovering new inhibitors of the GIRK1/4 channel UNIVERSITY OF SOUTH CAROLINA (US) 2012-12-04 US disclosed
US-20110281278-A1 High Throughput Assay for Discovering New Inhibitors of the GIRK1/4 Channel UNIVERSITY OF SOUTH CAROLINA (US) 2011-11-17 US disclosed