SCHEMBL13308397

SCHEMBL13308397

Cc1cc(-c2c(C)nn(Cc3cccc(C(F)(F)F)c3)c2C)ccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
ABHD6 Q9BV23 1/20 0.41
AR P10275 4/20 0.40
PTGDR2 Q9Y5Y4 3/20 0.39
TEC P42680 1/20 0.39
TXK P42681 1/20 0.39
BMX P51813 1/20 0.39
BTK Q06187 1/20 0.39
KCNK3 O14649 1/20 0.38
CNR1 P21554 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
P2RY14 Q15391 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3070135 0.90 HTT (0.46) POLBHTTL3MBTL1GRIN1GRIN2B
SCHEMBL13308563 0.86 EGLN2 (0.39) POLBHTTL3MBTL1ARGAA
SCHEMBL13308971 0.82 CYP1A2 (0.43) HTTARGAAMAPT
SCHEMBL3084002 0.82 AR (0.48) L3MBTL1GRIN1GRIN2BAR
SCHEMBL13309099 0.81 FNTA (0.43) POLBARGAANPSR1
SCHEMBL13308619 0.81 POLB (0.45) POLBARPTGDR2GAANPSR1
SCHEMBL3076403 0.80 AR (0.47) ARPTGDR2
SCHEMBL13309112 0.80 MBOAT4 (0.39) ARCNR1
SCHEMBL3085333 0.79 AR (0.42) POLBHTTL3MBTL1AR
SCHEMBL3069365 0.79 AR (0.48) ARPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194045-A1 SUBSTITUTED PYRAZOLE DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2010-06-09 EP disclosed