SCHEMBL13314766

SCHEMBL13314766

CC(C)(C)[C@H]1CCCc2sc(NC(=N)N)nc21

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
PSEN1 P49768 7/20 0.33
PSEN2 P49810 7/20 0.33
APH1B Q8WW43 7/20 0.33
NCSTN Q92542 7/20 0.33
APH1A Q96BI3 7/20 0.33
PSENEN Q9NZ42 7/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.33
MAPT P10636 1/20 0.31
XIAP P98170 2/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
PI4KB Q9UBF8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3542463 1.00 NPC1 (0.33) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL13314780 0.82 NPC1 (0.35) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3535415 0.82 NPC1 (0.35) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3536165 0.77 NPC1 (0.34) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3536663 0.77 NPC1 (0.34) NPC1RAB9APSEN1PSEN2APH1B
Formic Acid SCHEMBL3536155 0.77 TSHR (0.34) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3536953 0.76 XIAP (0.36) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL13349056 0.76 NPC1 (0.33) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL20000890 0.76 XIAP (0.32) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3538767 0.76 PSEN1 (0.33) NPC1RAB9APSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727979-B2 Guanidine derivatives and their use as neuropeptide FF receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2010-06-01 US disclosed
US-7727979-B2 Guanidine derivatives and their use as neuropeptide FF receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2010-06-01 US disclosed