SCHEMBL13325201

SCHEMBL13325201

CCc1ccc(C[C@@H](NC(=O)N2CCC(NCCc3ccccc3N)CC2)C(=O)N2CCC(N3CCCN(C)CC3)CC2)cc1CC

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 16/20 0.46
CYP3A4 P08684 11/20 0.45
CALCA P06881 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13325968 0.97 CALCRL (0.46) CALCRLCYP3A4CALCA
SCHEMBL13325991 0.96 CALCRL (0.49) CALCRLCYP3A4CALCA
SCHEMBL13326278 0.94 CALCRL (0.52) CALCRLCYP3A4CALCA
SCHEMBL13325959 0.94 CALCRL (0.52) CALCRLCYP3A4CALCA
SCHEMBL13325975 0.91 CALCRL (0.44) CALCRLCYP3A4CALCA
SCHEMBL13404720 0.90 CALCRL (0.44) CALCRLCYP3A4CALCA
SCHEMBL13326277 0.90 CALCRL (0.44) CALCRLCYP3A4CALCA
SCHEMBL13325727 0.90 CALCRL (0.46) CALCRLCYP3A4CALCA
SCHEMBL13325218 0.89 CALCRL (0.44) CALCRLCYP3A4CALCA
SCHEMBL13325726 0.89 CALCRL (0.46) CALCRLCYP3A4CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100152171-A1 CGRP Antagonists BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2010-06-17 US disclosed
US-7700589-B2 CGRP antagonists BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2010-04-20 US disclosed
US-20070244099-A1 CGRP Antagonists RUDOLF KLAUS 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070244099-A1 CGRP Antagonists CALCRL, OPRL1, CALCA CALCRL 1/4885CYP3A4 2631/4885CALCA 3/4885
US-20100152171-A1 CGRP Antagonists CALCRL, OPRL1, CALCA CALCRL 1/4885CYP3A4 2631/4885CALCA 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.