SCHEMBL13330583

SCHEMBL13330583

CC(F)(F)c1cc(Cl)c2nc(-c3nnc(-c4ccccc4Cl)o3)cn2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.50
RAB9A P51151 9/20 0.50
SMN1; SMN2 Q16637 7/20 0.50
NFKB1 P19838 6/20 0.50
NFKB2 Q00653 6/20 0.50
RELA Q04206 6/20 0.50
MAPT P10636 5/20 0.50
TP53 P04637 4/20 0.46
HPGD P15428 3/20 0.46
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RECQL P46063 1/20 0.44
KDM4E B2RXH2 6/20 0.43
ALDH1A1 P00352 6/20 0.43
PKM P14618 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340587 0.91 NPC1 (0.61) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13330828 0.84 NPC1 (0.46) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13331059 0.76 NPC1 (0.37) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13331095 0.75 SMN1; SMN2 (0.36) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3345955 0.75 NPC1 (0.60) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3338543 0.75 NPC1 (0.60) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3341804 0.75 SMN1; SMN2 (0.57) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3341149 0.74 SMN1; SMN2 (0.50) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3339342 0.74 RAB9A (0.53) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL3340937 0.74 NPC1 (0.45) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065760-A1 IMIDAZO [1,2A] PYRIDINE DERIVATIVES, THEIR USE AS S1P1 AGONISTS AND METHODS FOR THEIR PRODUCTION EXELIXIS, INC. (US) 2010-06-10 WO disclosed