SCHEMBL13344249

SCHEMBL13344249

CC1(C)CCc2c(-c3nc(-c4ccc(C=O)cc4)no3)n[nH]c2C1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALPL P05186 3/20 0.33
ITK Q08881 2/20 0.33
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
BRD4 O60885 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPT P10636 4/20 0.31
HPGD P15428 1/20 0.30
HSD11B1 P28845 1/20 0.30
AURKA O14965 1/20 0.30
LCK P06239 1/20 0.30
TP53 P04637 1/20 0.30
S1PR1 P21453 2/20 0.30
S1PR3 Q99500 2/20 0.30
AHR P35869 1/20 0.30
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3462090 0.79 S1PR1 (0.38) ITKS1PR1S1PR3
SCHEMBL13263031 0.77 S1PR1 (0.44) ITKAURKAS1PR1S1PR3
SCHEMBL30629157 0.77 RIPK1 (0.32) ITKRIPK1
SCHEMBL30629099 0.77 ITK (0.34) ITKMEN1KMT2AMAPTHPGD
SCHEMBL2476418 0.76 S1PR1 (0.36) ITKS1PR1S1PR3
SCHEMBL2543824 0.76 S1PR1 (0.36) NPC1RAB9AMAPTHSD11B1TP53
SCHEMBL13262772 0.75 S1PR1 (0.43) ITKS1PR1S1PR3
SCHEMBL1861990 0.73 S1PR1 (0.55) NPC1RAB9AMAPTTP53S1PR1
SCHEMBL13262879 0.71 S1PR1 (0.38) ALPLITKS1PR1S1PR3
SCHEMBL2470310 0.71 S1PR1 (0.43) ITKS1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2202232-A1 1,2,4-oxadiazole derivatives and their therapeutic use Laboratorios Almirall, S.A. (ES) 2010-06-30 EP disclosed