SCHEMBL13345657

SCHEMBL13345657

CCCC(C)Nc1ccc(-c2nc(-c3ccc4c(c3)CN(CCC(=O)O)CC4)no2)cc1C(F)(F)F

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.65
S1PR3 Q99500 7/20 0.55
S1PR5 Q9H228 2/20 0.46
S1PR4 O95977 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2168613 0.81 S1PR1 (0.84) S1PR1S1PR3S1PR5
SCHEMBL2417428 0.79 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL2181741 0.78 S1PR1 (0.79) S1PR1S1PR3S1PR5S1PR4CYP2C9
SCHEMBL2179933 0.78 S1PR1 (0.79) S1PR1S1PR3S1PR5S1PR4CYP2C9
SCHEMBL2420104 0.77 S1PR1 (1.00) S1PR1S1PR3S1PR5S1PR4CYP2C9
Trifluoroacetic Acid SCHEMBL1870072 0.75 S1PR1 (0.61) S1PR1S1PR3S1PR5S1PR4CYP2C9
SCHEMBL2484873 0.74 S1PR1 (0.88) S1PR1S1PR3S1PR5
SCHEMBL2169176 0.74 S1PR1 (0.73) S1PR1S1PR3
SCHEMBL2994820 0.74 S1PR1 (0.75) S1PR1S1PR3S1PR5CYP2C9
SCHEMBL16659635 0.73 S1PR1 (0.90) S1PR1S1PR3S1PR5S1PR4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069949-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS MERCK SERONO S.A. (CH) 2010-06-24 WO disclosed