SCHEMBL2484873

SCHEMBL2484873

Cc1ccccc1-c1ccc(-c2nc(-c3ccc4c(c3)CN(CCC(=O)O)CC4)no2)cc1C(F)(F)F.Cc1ccccc1-c1ccc(-c2nc(-c3ccc4c(c3)CN(CCC(=O)OC(C)(C)C)CC4)no2)cc1C(F)(F)F

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.88
S1PR3 Q99500 3/20 0.50
S1PR5 Q9H228 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2416941 0.97 S1PR1 (0.82) S1PR1S1PR3S1PR5
SCHEMBL2417428 0.94 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL3467816 0.90 S1PR1 (0.82) S1PR1S1PR3
SCHEMBL2485876 0.89 S1PR1 (0.88) S1PR1S1PR3S1PR5
SCHEMBL4746452 0.88 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL2413715 0.86 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL2168613 0.85 S1PR1 (0.84) S1PR1S1PR3S1PR5
SCHEMBL2420128 0.85 S1PR1 (0.83) S1PR1S1PR3S1PR5
SCHEMBL16659664 0.83 S1PR1 (0.90) S1PR1S1PR3
SCHEMBL2181741 0.82 S1PR1 (0.79) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376484-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS Merck Serono S.A. (CH) 2011-10-19 EP disclosed
WO-2010069949-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS MERCK SERONO S.A. (CH) 2010-06-24 WO disclosed