SCHEMBL13348703

SCHEMBL13348703

CN(C(=O)OC(C)(C)C)c1nc(N)c(C2CCCCC2)c2c1ncn2C

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.33
PIK3CD O00329 1/20 0.33
TNK2 Q07912 1/20 0.33
MAP4K4 O95819 3/20 0.32
CPB2 Q96IY4 1/20 0.32
CDK1 P06493 1/20 0.32
PDE8B O95263 1/20 0.31
BACE1 P56817 2/20 0.30
CTSD P07339 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2768416 0.83 MAP4K4 (0.31) IKBKBPIK3CDMAP4K4
SCHEMBL2767551 0.83 PAX8 (0.33) IKBKBPIK3CDMAP4K4CDK1
SCHEMBL3880903 0.82 CDK1 (0.34) MAP4K4CDK1
SCHEMBL2768343 0.82 CSF1R (0.38) IKBKB
SCHEMBL12344427 0.79 CDK1 (0.36) IKBKBCDK1
SCHEMBL12344385 0.78 BRD4 (0.38) IKBKB
SCHEMBL12341871 0.75 GRM4 (0.32)
SCHEMBL13463910 0.74 BRD4 (0.39) IKBKBTNK2
SCHEMBL12344450 0.74 IKBKB (0.32) IKBKB
SCHEMBL12344495 0.74 FNTA (0.37) IKBKBMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7737279-B2 1,6-dihydro-1,3,5,6-tetraaza-as-indacene based tricyclic compounds and pharmaceutical compositions comprising same BRISTOL-MYERS SQUIBB COMPANY (US) 2010-06-15 US disclosed