SCHEMBL13360729

SCHEMBL13360729

CCOOCC1=C(NC(=O)NC(c2ccccc2)c2ccccc2)CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.39
ESR2 Q92731 1/20 0.39
MAPK1 P28482 1/20 0.38
GPR119 Q8TDV5 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
GLS O94925 1/20 0.36
BACE1 P56817 1/20 0.36
NAMPT P43490 1/20 0.36
NR1H2 P55055 1/20 0.36
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 2/20 0.35
ALOX15 P16050 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HTT P42858 1/20 0.35
PTGER4 P35408 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13271789 0.85 ATM (0.37) ATMESR2MAPK1GPR119HDAC1
SCHEMBL13329601 0.83 ADORA1 (0.41) ATMMAPK1GPR119GLSTSHR
SCHEMBL13271560 0.76 GPR119 (0.48) ESR2GPR119HDAC1HDAC6GLS
SCHEMBL13329617 0.75 NPY2R (0.41) ATMMAPK1GLSTSHRMEN1
SCHEMBL13250469 0.73 NPY2R (0.41) ATMMAPK1TSHRMEN1KMT2A
SCHEMBL13360730 0.72 ESR2 (0.50) ESR2MAPK1NR1H2KDM4E
SCHEMBL13271559 0.70 ADORA1 (0.47) ESR2MAPK1NR1H2KDM4E
SCHEMBL21047249 0.69 ADORA1 (0.43) ATMESR2GPR119GLSTSHR
SCHEMBL1219803 0.69 ADORA1 (0.43) ATMESR2GPR119GLSTSHR
SCHEMBL1219800 0.69 ADORA1 (0.43) ATMESR2GPR119GLSTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130584-A1 PYRIMIDINONE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2008-10-30 WO disclosed