SCHEMBL1336727

SCHEMBL1336727

CC(C)(C)OC(=O)N1C[C@@H](F)C[C@H]1C(=O)N[C@H]1CC[C@@H]2CNC[C@@H]21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.32
CTSL P07711 2/20 0.32
CTSB P07858 2/20 0.32
CTSS P25774 2/20 0.32
CTSK P43235 2/20 0.32
HTRA1 Q92743 1/20 0.32
USP30 Q70CQ3 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
HSD11B1 P28845 1/20 0.30
NR1H2 P55055 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1336138 1.00 CYP1A2 (0.34) CYP1A2POLBCYP3A4CYP2C19SMN1; SMN2
SCHEMBL1336140 1.00 CYP1A2 (0.34) CYP1A2POLBCYP3A4CYP2C19SMN1; SMN2
SCHEMBL16498240 1.00 CYP1A2 (0.34) CYP1A2POLBCYP3A4CYP2C19SMN1; SMN2
SCHEMBL16498034 0.83 CFD (0.32) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL16498621 0.76 CACNA1B (0.41) HTRA1
SCHEMBL1336730 0.76 CACNA1B (0.41) HTRA1
SCHEMBL1336728 0.76 CACNA1B (0.41) HTRA1
SCHEMBL18610727 0.74 PTPN1 (0.44) CYP1A2POLBCYP3A4CYP2C19SMN1; SMN2
SCHEMBL1337445 0.73 CACNA1B (0.53) NR1H2
SCHEMBL18849689 0.73 CYP1A2 (0.42) CYP1A2POLBCYP3A4CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110281870-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA[C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110281870-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA[C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS CACNA1C, ORAI1, CACNA1S CYP1A2 545/4885POLB 3123/4885CYP3A4 1006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.