SCHEMBL13368199

SCHEMBL13368199

CCCN1C(=O)C(C)(C)c2cc3[nH]c(CCc4ccccc4)nc3cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.46
AURKB Q96GD4 1/20 0.46
RAB9A P51151 3/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
NPC1 O15118 1/20 0.43
HDAC6 Q9UBN7 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13341279 0.93 AURKA (0.44) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2488708 0.87 AURKA (0.40) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2511374 0.86 AURKA (0.43) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2492165 0.86 AURKA (0.43) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2488713 0.86 AURKA (0.43) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2488719 0.86 AURKA (0.43) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL3424599 0.85 HDAC1 (0.41) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL13341319 0.84 HDAC6 (0.45) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL2486444 0.84 MAPT (0.45) AURKAAURKBRAB9AMAPTSMN1; SMN2
SCHEMBL3426661 0.84 RAB9A (0.48) RAB9AMAPTSMN1; SMN2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714010-B2 Pyrrolobenzimidazolones and their use as anti-proliferative agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-11 US disclosed