SCHEMBL13373301

SCHEMBL13373301

CCNc1ncc2c(n1)-c1nc(C)sc1CO2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 10/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
CYP1A2 P05177 9/20 0.33
HSD17B10 Q99714 9/20 0.33
CASP1 P29466 7/20 0.33
CASP7 P55210 7/20 0.33
CLK4 Q9HAZ1 5/20 0.33
USP2 O75604 5/20 0.33
TSHR P16473 4/20 0.33
MAPK1 P28482 3/20 0.33
GLA P06280 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP3A4 P08684 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13373400 0.86 ALDH1A1 (0.33) GAAL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL13373297 0.81 CCNE1 (0.40) ALDH1A1MEN1KMT2ACYP1A2HSD17B10
SCHEMBL13373339 0.81 ALDH1A1 (0.32) GAAALDH1A1MEN1KMT2ACYP1A2
SCHEMBL13373284 0.80 ADORA2A (0.32) GAAL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL13373271 0.78 ALDH1A1 (0.32) GAAL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL13373340 0.77 ADORA1 (0.37) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL13373279 0.76 CDK2 (0.42) ALDH1A1MEN1KMT2ACYP1A2HSD17B10
SCHEMBL13373311 0.75 ALDH1A1 (0.33) GAAALDH1A1MEN1KMT2ACYP1A2
SCHEMBL13373283 0.74 CCNE1 (0.33) GAAALDH1A1MEN1KMT2ACYP1A2
SCHEMBL13373382 0.74 ALDH1A1 (0.36) GAAALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8288400-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-16 US disclosed