SCHEMBL13385183

SCHEMBL13385183

Cc1ccc(Oc2nc3cc(-c4ccc5c(c4)CNC5=O)c(Cl)cc3[nH]2)cc1C=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 14/20 0.51
PRKAB1 Q9Y478 14/20 0.51
PRKAA2 P54646 11/20 0.51
PRKAA1 Q13131 6/20 0.51
PRKAB2 O43741 1/20 0.51
TFDP2 Q14188 1/20 0.51
PRKAG3 Q9UGI9 1/20 0.51
PRKAG2 Q9UGJ0 1/20 0.51
DAPK3 O43293 1/20 0.37
NTRK1 P04629 1/20 0.37
PIM1 P11309 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
ROCK1 Q13464 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
CHEK2 O96017 2/20 0.36
MAPKAPK2 P49137 1/20 0.36
BRAF P15056 1/20 0.35
AURKA O14965 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3481056 0.86 PRKAG1 (0.71) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL3481238 0.78 PRKAG1 (0.69) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL3481068 0.73 PRKAG1 (0.72) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL13402925 0.72 PRKAG1 (0.74) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL19312548 0.71 PRKAG1 (0.50) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL3481411 0.71 PRKAG1 (0.71) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL3481222 0.70 PRKAG1 (0.72) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL13403018 0.70 PRKAG1 (0.84) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL823781 0.70 PRKAG1 (0.78) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2
SCHEMBL13402923 0.69 PRKAG1 (0.72) PRKAG1PRKAB1PRKAA2PRKAA1PRKAB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036613-A1 NOVEL CYCLIC BENZIMIDAZOLE DERIVATIVES USEFUL ANTI-DIABETIC AGENTS MERCK SHARP & DOHME CORP. (US) 2010-04-01 WO disclosed