SCHEMBL13385682

SCHEMBL13385682

CC(C)(CC(CC(=O)c1ccc(C(F)(F)F)cc1)c1ccc(Cl)cc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.46
POLB P06746 2/20 0.45
UTS2R Q9UKP6 2/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HSP90AA1 P07900 1/20 0.45
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CNR2 P34972 1/20 0.42
KMT2A Q03164 1/20 0.41
PTPN1 P18031 2/20 0.41
GSK3B P49841 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
FFAR1 O14842 3/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13385708 0.89 PDPK1 (0.59) PDPK1CYP2C9CYP2C19PTPN1GSK3B
SCHEMBL13385524 0.85 POLB (0.47) PDPK1POLBALDH1A1LMNAHSP90AA1
SCHEMBL13385550 0.84 CYP2C9 (0.62) PDPK1POLBALDH1A1LMNAHSP90AA1
SCHEMBL657017 0.84 GABBR2 (0.52) PDPK1POLBUTS2RLMNATHRB
SCHEMBL13385520 0.78 POLB (0.52) PDPK1POLBUTS2RALDH1A1LMNA
SCHEMBL657567 0.76 PDPK1 (0.78) PDPK1POLBUTS2RALDH1A1LMNA
SCHEMBL19320567 0.75 CYP1A2 (0.45) LMNAMAPTTHRBCYP2C9CYP2C19
SCHEMBL12174638 0.73 PDPK1 (0.57) PDPK1POLBNPSR1CYP2C9CYP2C19
SCHEMBL28818751 0.73 PDPK1 (0.57) PDPK1POLBNPSR1CYP2C9CYP2C19
SCHEMBL28818750 0.73 PDPK1 (0.57) PDPK1POLBNPSR1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed