SCHEMBL13401477

SCHEMBL13401477

O=Cc1ccc(NC(=O)c2cc(F)ccc2F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.54
RAB9A P51151 6/20 0.52
NPC1 O15118 5/20 0.52
TDP1 Q9NUW8 2/20 0.52
CTDSP1 Q9GZU7 1/20 0.52
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
SNCA P37840 2/20 0.49
P2RX1 P51575 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
GRM5 P41594 1/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
KLK7 P49862 1/20 0.44
LCLAT1 Q6UWP7 1/20 0.44
FADS1 O60427 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8859383 0.85 SMN1; SMN2 (0.50) LMNARAB9ANPC1TDP1CTDSP1
SCHEMBL6816710 0.81 LMNA (0.57) LMNARAB9ANPC1TDP1CTDSP1
SCHEMBL24023021 0.79 LMNA (0.58) LMNARAB9ANPC1TDP1KMT2A
SCHEMBL14185647 0.79 P2RX1 (0.48) LMNARAB9ANPC1TDP1KMT2A
SCHEMBL8126465 0.78 HTT (0.67) LMNAKMT2AMEN1HTTMAPT
SCHEMBL6593406 0.78 PTPN1 (0.69) RAB9ANPC1TDP1KMT2AMEN1
SCHEMBL18160397 0.75 LMNA (0.61) LMNARAB9ANPC1TDP1CTDSP1
SCHEMBL18146857 0.75 LMNA (0.61) LMNARAB9ANPC1TDP1KMT2A
SCHEMBL19873379 0.75 LMNA (0.61) LMNARAB9ANPC1TDP1KMT2A
SCHEMBL7081255 0.74 LMNA (0.49) LMNARAB9ANPC1TDP1CTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7691844-B2 Nonpeptide substituted spirobenzoazepines as vasopressin antagonists ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2010-04-06 US disclosed