SCHEMBL13406478

SCHEMBL13406478

C[C@H]1CNCC[C@H]1c1ccc(F)c(C(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 1/20 0.45
AKT1 P31749 8/20 0.40
AKT2 P31751 3/20 0.40
SGK1 O00141 2/20 0.40
RPS6KB1 P23443 2/20 0.40
PRKCQ Q04759 2/20 0.40
ROCK1 Q13464 2/20 0.40
RPS6KA1 Q15418 2/20 0.40
AKT3 Q9Y243 2/20 0.40
ROCK2 O75116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13406473 1.00 P2RY14 (0.45) P2RY14AKT1AKT2SGK1RPS6KB1
SCHEMBL13406477 1.00 P2RY14 (0.45) P2RY14AKT1AKT2SGK1RPS6KB1
SCHEMBL13406479 1.00 P2RY14 (0.45) P2RY14AKT1AKT2SGK1RPS6KB1
SCHEMBL13406376 0.86 ALDH1A1 (0.44) AKT1AKT2SGK1RPS6KB1PRKCQ
SCHEMBL3624844 0.86 ALDH1A1 (0.44) AKT1AKT2SGK1RPS6KB1PRKCQ
SCHEMBL13645918 0.86 ALDH1A1 (0.44) AKT1AKT2SGK1RPS6KB1PRKCQ
SCHEMBL13646126 0.85 P2RY14 (0.44) P2RY14
SCHEMBL13646123 0.85 P2RY14 (0.44) P2RY14
SCHEMBL13646125 0.85 P2RY14 (0.44) P2RY14
SCHEMBL13646124 0.85 P2RY14 (0.44) P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700591-B2 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors MERCK & CO., INC. (US) 2010-04-20 US disclosed
US-7700591-B2 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors MERCK & CO., INC. (US) 2010-04-20 US disclosed