SCHEMBL13407672

SCHEMBL13407672

CN1C(=N)N[C@](CCC2CCCCC2)(CC2CCC[C@@H](Nc3ccc4ccccc4n3)C2)C1=O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.56
CTSD P07339 14/20 0.56
MCHR1 Q99705 1/20 0.42
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7546165 1.00 BACE1 (0.56) BACE1CTSDMCHR1DDB1CRBN
SCHEMBL8411137 0.92 BACE1 (0.48) BACE1CTSDMCHR1DDB1CRBN
SCHEMBL7541503 0.90 CTSD (0.47) BACE1CTSDMCHR1DDB1CRBN
SCHEMBL8412199 0.90 BACE1 (0.48) BACE1CTSDMCHR1DDB1CRBN
SCHEMBL7536828 0.90 BACE1 (0.46) BACE1CTSDMCHR1
SCHEMBL13407674 0.90 BACE1 (0.57) BACE1CTSDPRMT5WDR77
SCHEMBL7538807 0.90 BACE1 (0.57) BACE1CTSDPRMT5WDR77
SCHEMBL7540242 0.89 BACE1 (0.45) BACE1CTSDMCHR1
SCHEMBL8412486 0.88 BACE1 (0.44) BACE1CTSDMCHR1
SCHEMBL7539290 0.88 MCHR1 (0.48) BACE1CTSDMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700603-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-04-20 US disclosed
US-7700603-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-04-20 US disclosed