SCHEMBL13409353

SCHEMBL13409353

COc1cc2ccnc(OC(C)C)c2cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
TRPA1 O75762 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
TNF P01375 3/20 0.42
ACHE P22303 3/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
IRAK4 Q9NWZ3 2/20 0.39
SRC P12931 1/20 0.39
KMO O15229 1/20 0.38
PDE10A Q9Y233 3/20 0.38
USP2 O75604 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 2/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13409354 0.83 TRPA1 (0.58) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL8271696 0.82 TRPA1 (0.51) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL8273097 0.81 MEN1 (0.48) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL1536597 0.79 TNF (0.48) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL13409326 0.76 ATM (0.40) TNFL3MBTL1IRAK4MAPT
SCHEMBL13409741 0.75 TNF (0.49) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL13385161 0.75 TRPA1 (0.56) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL13409340 0.74 CYP19A1 (0.43) TRPA1CYP2C19TRPM8L3MBTL1KMO
SCHEMBL24250119 0.72 IRAK4 (0.45) CYP3A4TRPA1CYP1A2CYP2D6CYP2C9
SCHEMBL13409343 0.71 LRRK2 (0.42) CYP1A2IRAK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7705146-B2 Hepatitis C inhibitor peptide analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-27 US disclosed