SCHEMBL13420656

SCHEMBL13420656

Bc1cnc(Nc2cc(Cl)cc(OC)c2)nc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.43
FGFR1 P11362 2/20 0.43
HDAC3 O15379 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
BRD4 O60885 1/20 0.42
PLK1 P53350 1/20 0.41
IGF1R P08069 2/20 0.40
SYK P43405 4/20 0.40
SRC P12931 1/20 0.38
ZAP70 P43403 1/20 0.38
PIK3CA P42336 3/20 0.38
PIK3CB P42338 3/20 0.38
PIK3CG P48736 3/20 0.38
CDK2 P24941 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK5 Q00535 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13420657 0.88 JAK2 (0.44) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL3448950 0.84 IGF1R (0.51) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL3448147 0.76 IGF1R (0.49) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL3345672 0.76 IGF1R (0.57) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL13421116 0.74 HDAC3 (0.46) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL23021288 0.74 PLK1 (0.47) EGFRFGFR1HDAC3HDAC1HDAC2
Hydrochloric Acid SCHEMBL22999798 0.73 PLK1 (0.46) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL3450370 0.72 IGF1R (0.53) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL13420648 0.71 HDAC3 (0.50) EGFRFGFR1HDAC3HDAC1HDAC2
SCHEMBL20752152 0.69 LRRK2 (0.61) BRD4IGF1RJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed