SCHEMBL13423939

SCHEMBL13423939

C=C1CCn2nc(NC(C)=O)cc2C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.37
ADORA1 P30542 5/20 0.37
MAP4K4 O95819 1/20 0.37
ABL1 P00519 1/20 0.37
MAPK8 P45983 1/20 0.37
CSNK1A1 P48729 1/20 0.37
CDK7 P50613 1/20 0.37
TYRO3 Q06418 1/20 0.37
LRRK2 Q5S007 1/20 0.37
AURKB Q96GD4 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
PIK3CG P48736 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
AOC3 Q16853 2/20 0.36
PIK3C3 Q8NEB9 2/20 0.34
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15477979 0.78 MAP4K4 (0.36) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423899 0.77 CYP1A2 (0.41) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423938 0.76 ADORA2A (0.38) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL15477976 0.74 ADORA2A (0.35) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13424078 0.69 DRD4 (0.36) MAP4K4ABL1MAPK8CSNK1A1CDK7
SCHEMBL13423946 0.67 PIK3C3 (0.34) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423883 0.65 ADORA1 (0.44) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423902 0.65 DRD4 (0.39) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423903 0.64 NR3C2 (0.39) ADORA2AADORA1MAP4K4ABL1MAPK8
SCHEMBL13423905 0.64 WNT3A (0.40) ADORA2AADORA1MAP4K4ABL1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043676-A1 TETRA-AZA-HETEROCYCLES AS PHOSPHATIDYLINOSITOL-3-KINASES (PI3-KINASES) INHIBITOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-22 WO disclosed