SCHEMBL13423978

SCHEMBL13423978

COC(=O)c1ccc2[nH]c(-c3ccc(N(C)O)cc3)c(-c3ccccc3)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
FLT3 P36888 1/20 0.50
KIF11 P52732 1/20 0.48
PTGS2 P35354 7/20 0.46
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
MDH2 P40926 1/20 0.44
GSK3B P49841 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 1/20 0.43
PPARG P37231 1/20 0.42
GPR84 Q9NQS5 1/20 0.42
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2285692 0.90 MEN1 (0.71) MEN1KMT2AFLT3KIF11PTGS2
SCHEMBL2290102 0.82 MEN1 (0.58) MEN1KMT2AFLT3KIF11PTGS2
SCHEMBL2818000 0.76 MEN1 (0.56) MEN1KMT2AFLT3KIF11CCNB2
SCHEMBL2284207 0.76 PPARG (0.63) MEN1KMT2AFLT3PTGS2KDM4E
SCHEMBL29031872 0.76 PARP1 (0.59) MEN1KMT2AFLT3KIF11CCNB2
SCHEMBL30472344 0.76 PARP1 (0.59) MEN1KMT2AFLT3KIF11CCNB2
SCHEMBL10746161 0.75 MEN1 (0.57) MEN1KMT2AFLT3KIF11CCNB2
SCHEMBL5441431 0.74 MEN1 (0.54) MEN1KMT2AFLT3KIF11CCNB2
SCHEMBL7040925 0.74 ESR1 (0.68) MEN1KMT2AFLT3KIF11PTGS2
SCHEMBL11558711 0.74 MEN1 (0.69) MEN1KMT2AFLT3KIF11CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046013-A1 AZAINDOLE DERIVATIVE MERCK PATENT GMBH (DE) 2010-04-29 WO disclosed