SCHEMBL13425243

SCHEMBL13425243

NC1=NC=NC2C1C(c1ccc(O)nc1)=NN2Cc1cc2ccccc2nc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 4/20 0.40
PIK3C2B O00750 2/20 0.39
PIK3CG P48736 8/20 0.38
MYC P01106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425242 0.89 PIK3CD (0.48) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425239 0.89 PIK3CD (0.43) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425246 0.89 PIK3CD (0.41) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425221 0.83 PIK3CD (0.54) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425212 0.76 PIK3CG (0.48) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425245 0.75 PIK3CD (0.41) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425087 0.70 PIK3C2B (0.53) PIK3CDPIK3C2BPIK3CG
SCHEMBL13424912 0.70 PIK3CD (0.55) PIK3CDPIK3C2BPIK3CG
SCHEMBL682419 0.69 PIK3C2B (0.72) PIK3CDPIK3C2BPIK3CG
SCHEMBL13425086 0.69 PIK3CD (0.40) PIK3CDPIK3C2BPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9790228-B2 Heterocyclic kinase inhibitors INTELLIKINE LLC (US) 2017-10-17 US disclosed
US-9790228-B2 Heterocyclic kinase inhibitors INTELLIKINE LLC (US) 2017-10-17 US disclosed
US-20160168157-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE LLC 2016-06-16 US disclosed
US-20160168157-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE LLC 2016-06-16 US disclosed
WO-2010036380-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE, INC. (US) 2010-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160168157-A1 HETEROCYCLIC KINASE INHIBITORS MAP3K13, MAP3K3, CDK3 PIK3CD 147/4885PIK3C2B 132/4885PIK3CG 191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.