SCHEMBL13430255

SCHEMBL13430255

COc1cc2ncnc(NCCC3CN=C(NC(=O)Nc4cccc(Br)c4)S3)c2cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.61
EGFR P00533 8/20 0.61
KIT P10721 2/20 0.61
AURKA O14965 2/20 0.53
SRC P12931 2/20 0.53
RAF1 P04049 1/20 0.53
MET P08581 1/20 0.53
PDGFRB P09619 1/20 0.53
FLT1 P17948 1/20 0.53
FLT4 P35916 1/20 0.53
ERBB2 P04626 2/20 0.51
FBP1 P09467 2/20 0.51
KDM4E B2RXH2 1/20 0.51
GAK O14976 1/20 0.51
MAPK13 O15264 1/20 0.51
ABL1 P00519 1/20 0.51
CYP1A2 P05177 1/20 0.51
CDK1 P06493 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13430289 0.91 EGFR (0.56) KDREGFRKITAURKASRC
SCHEMBL13430229 0.84 AURKA (0.56) KDREGFRAURKAERBB2HDAC3
SCHEMBL13399987 0.77 AURKA (0.83) KDREGFRKITAURKASRC
SCHEMBL31067695 0.76 KDR (1.00) KDREGFRKITSRCRAF1
SCHEMBL13430282 0.75 AURKA (0.44) KDREGFRAURKAFLT1FLT4
SCHEMBL13429852 0.75 MAP2K1 (0.50) KDREGFRSRCRAF1FLT1
SCHEMBL13430228 0.74 AURKA (0.69) KDREGFRAURKA
SCHEMBL13430238 0.74 AURKA (0.56) EGFRAURKAKDM4E
SCHEMBL13430283 0.74 AURKA (0.54) KDREGFRAURKAKDM4E
SCHEMBL13430199 0.74 AURKA (0.64) KDREGFRKITAURKAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036629-A2 FUSED MULTICYCLIC COMPOUNDS AS PROTEIN KINASE INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2010-04-01 WO disclosed