SCHEMBL13430282

SCHEMBL13430282

COc1cc2ncnc(NCCC3CN=C(NC(=O)Nc4ccccc4)S3)c2nc1OCCN(C)C

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKA O14965 12/20 0.44
KDR P35968 6/20 0.41
AURKB Q96GD4 2/20 0.40
EGFR P00533 4/20 0.39
CSF1R P07333 1/20 0.38
BRAF P15056 1/20 0.37
RPS6KB1 P23443 1/20 0.37
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13429732 0.91 AURKA (0.46) AURKAKDRAURKBEGFRCSF1R
SCHEMBL13430229 0.84 AURKA (0.56) AURKAKDRAURKBEGFR
SCHEMBL13399874 0.81 AURKA (0.69) AURKAKDRAURKBCSF1RRPS6KB1
SCHEMBL13430228 0.78 AURKA (0.69) AURKAKDRAURKBEGFRCSF1R
SCHEMBL13430278 0.78 AURKA (0.38) AURKAKDRAURKBEGFRCSF1R
SCHEMBL13430283 0.78 AURKA (0.54) AURKAKDRAURKBEGFRCSF1R
SCHEMBL13430238 0.77 AURKA (0.56) AURKAAURKBEGFRCSF1R
SCHEMBL13430271 0.76 AURKA (0.48) AURKAAURKBCSF1RRPS6KB1
SCHEMBL13430281 0.75 AURKA (0.49) AURKAAURKBCSF1RRPS6KB1
SCHEMBL13430255 0.75 KDR (0.61) AURKAKDREGFRFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8765953-B2 Compounds and methods for the treatment of pain and other diseases AQUILUS PHARMACEUTICALS, INC. (US) 2014-07-01 US disclosed
WO-2010036629-A2 FUSED MULTICYCLIC COMPOUNDS AS PROTEIN KINASE INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2010-04-01 WO disclosed