SCHEMBL1343080

SCHEMBL1343080

Cc1ccc(NC(=O)C(=O)Nc2nc(CNS(C)(=O)=O)cs2)c(C(=O)C2CCCC2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 2/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.37
ALDH1A1 P00352 2/20 0.36
ABCC1 P33527 1/20 0.36
TYR P14679 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ATAD2 Q6PL18 1/20 0.34
ACKR3 P25106 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1342591 0.92 SMN1; SMN2 (0.39) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL1342825 0.89 RAB9A (0.45) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL6692815 0.89 AVPR1B (0.42) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL1340437 0.85 SMN1; SMN2 (0.36) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL2666123 0.85 GAA (0.47) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL1341610 0.84 TP53 (0.38) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL1341317 0.83 RAB9A (0.36) RAB9AKMT2ANPC1HTTMEN1
SCHEMBL1341936 0.83 CLK1 (0.37) RAB9AKMT2ANPC1HTTLMNA
SCHEMBL1341933 0.82 PIK3CD (0.36) KMT2AMEN1SMN1; SMN2GAAMAPT
SCHEMBL1342277 0.82 CLK1 (0.35) RAB9AKMT2ANPC1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063081-B2 N-(2-Phenoxyphenyl)-N'-(thiazol-2-yl)urea; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-11-22 US disclosed
US-7897628-B2 {2-[3-(4-Methyl-2-[2-methypropoxy]phenyl)-ureido]-thiazol-4-yl}-acetic acid ethyl ester; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-03-01 US disclosed
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents VTV THERAPEUTICS LLC 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents GCK, GCKR, PDK2 RAB9A 3353/4885KMT2A 1526/4885NPC1 2201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.