SCHEMBL13431990

SCHEMBL13431990

Nc1ccc(S(=O)(=O)N2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 17/20 1.00
PKLR P30613 8/20 0.82
NPC1 O15118 1/20 0.82
RAB9A P51151 1/20 0.82
MEN1 O00255 1/20 0.74
KMT2A Q03164 1/20 0.74
HTT P42858 2/20 0.72
LMNA P02545 2/20 0.69
KDM4E B2RXH2 1/20 0.69
ALDH1A1 P00352 1/20 0.69
TSHR P16473 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
CYP2C19 P33261 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12354636 0.96 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL1722758 0.91 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL15746503 0.87 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL1725568 0.87 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL1710857 0.85 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL1726834 0.85 PKM (1.00) PKMPKLRNPC1RAB9AMEN1
SCHEMBL30621219 0.84 PKM (1.00) PKMPKLRNPC1RAB9AHTT
SCHEMBL30621218 0.84 PKM (1.00) PKMPKLRNPC1RAB9AHTT
SCHEMBL12354635 0.84 PKM (1.00) PKMPKLRNPC1RAB9AHTT
SCHEMBL29483533 0.83 PKM (0.84) PKMPKLRNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042867-A2 ACTIVATORS OF HUMAN PYRUVATE KINASE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2010-04-15 WO disclosed