SCHEMBL1343399

SCHEMBL1343399

CC(C)COc1cc(F)ccc1NC(=O)C(=O)Nc1nc(CNS(C)(=O)=O)cs1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
MYC P01106 1/20 0.37
MAX P61244 1/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 2/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MKNK2 Q9HBH9 2/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1341682 0.92 GAA (0.40) SMN1; SMN2MAPTNPC1RAB9AKMT2A
SCHEMBL1342202 0.90 MYC (0.39) SMN1; SMN2MYCMAXMAPTNPC1
SCHEMBL1343578 0.89 GAA (0.43) SMN1; SMN2MAPTNPC1RAB9AKMT2A
SCHEMBL4461551 0.85 MAPT (0.44) SMN1; SMN2MYCMAXMAPTNPC1
SCHEMBL1342441 0.84 MKNK2 (0.36) MYCMAXMKNK2
SCHEMBL1342027 0.84 MKNK2 (0.36) MYCMAXMKNK2
SCHEMBL1343475 0.84 GCK (0.42) MYCMAXMKNK2
SCHEMBL1341627 0.84 GAA (0.43) SMN1; SMN2MAPTNPC1RAB9AKMT2A
SCHEMBL1342893 0.83 MKNK2 (0.36) MYCMAXMKNK2
SCHEMBL1340859 0.82 LPAR1 (0.39) MAPTNPC1KMT2ATP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063081-B2 N-(2-Phenoxyphenyl)-N'-(thiazol-2-yl)urea; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-11-22 US disclosed
US-7897628-B2 {2-[3-(4-Methyl-2-[2-methypropoxy]phenyl)-ureido]-thiazol-4-yl}-acetic acid ethyl ester; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-03-01 US disclosed
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents VTV THERAPEUTICS LLC 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents GCK, GCKR, PDK2 SMN1; SMN2 2958/4885MYC 180/4885MAX 2951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.