SCHEMBL13437152

SCHEMBL13437152

CC(C)(C)OC(=O)N1CCC(C(=O)NC2c3ccccc3-c3c(-c4nc5ccncc5[nH]4)cccc32)CC1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 5/20 0.60
PDE10A Q9Y233 1/20 0.41
PARP1 P09874 2/20 0.40
IDO1 P14902 3/20 0.40
CHEK2 O96017 1/20 0.39
GPR119 Q8TDV5 2/20 0.39
PDE5A O76074 2/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
FASN P49327 1/20 0.39
STS P08842 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
HASPIN Q8TF76 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12430894 0.75 HSP90AB1 (0.78) HSP90AB1PDE5AFASN
SCHEMBL13437168 0.74 HSP90AB1 (0.83) HSP90AB1PDE5A
SCHEMBL13437167 0.74 HSP90AB1 (0.85) HSP90AB1PDE5A
SCHEMBL13437191 0.74 HSP90AB1 (0.64) HSP90AB1PDE5A
SCHEMBL12430906 0.73 HSP90AB1 (0.78) HSP90AB1PDE5A
SCHEMBL12430459 0.72 HSP90AB1 (0.67) HSP90AB1PDE5A
SCHEMBL13437169 0.72 HSP90AB1 (0.81) HSP90AB1PDE5A
SCHEMBL13437213 0.71 HSP90AB1 (0.81) HSP90AB1PDE5A
SCHEMBL12430922 0.71 HSP90AB1 (0.79) HSP90AB1PDE5AFASN
SCHEMBL12430436 0.71 HSP90AB1 (0.70) HSP90AB1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7674795-B2 Fluorene derivatives, composition containing said derivatives and the use thereof AVENTIS PHARMA SA (FR) 2010-03-09 US disclosed
US-7674795-B2 Fluorene derivatives, composition containing said derivatives and the use thereof AVENTIS PHARMA SA (FR) 2010-03-09 US disclosed
US-20080153837-A1 Novel Fluorene Derivatives, Composition Containing Said Derivatives and the Use Thereof AVENTIS PHARMA S.A. (FR) 2008-06-26 US disclosed
US-20080153837-A1 Novel Fluorene Derivatives, Composition Containing Said Derivatives and the Use Thereof AVENTIS PHARMA S.A. (FR) 2008-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080153837-A1 Novel Fluorene Derivatives, Composition Containing Said Derivatives and the Use Thereof HSP90B1, HSP90AB1, HSP90AA1 HSP90AB1 2/4885PDE10A 3306/4885PARP1 2606/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.