SCHEMBL134430

SCHEMBL134430

COC(=O)NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C)cc1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
HTT P42858 1/20 0.58
POLB P06746 3/20 0.56
MAPT P10636 3/20 0.55
HSD17B10 Q99714 2/20 0.55
HPGD P15428 1/20 0.55
ALOX15 P16050 1/20 0.55
MAPK1 P28482 1/20 0.55
KDM4E B2RXH2 2/20 0.53
NPSR1 Q6W5P4 1/20 0.52
THRB P10828 1/20 0.52
NPC1 O15118 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897413 1.00 MEN1 (0.58) MEN1KMT2AHTTPOLBMAPT
SCHEMBL21225837 0.96 KMT2A (0.54) MEN1KMT2AHTTPOLBMAPT
SCHEMBL20601872 0.92 POLB (0.54) MEN1KMT2APOLBMAPTHSD17B10
SCHEMBL14809963 0.91 POLB (0.51) MEN1KMT2AHTTPOLBMAPT
Fluroxypyr SCHEMBL28706288 0.83 POLB (0.45) MEN1KMT2AHTTPOLBMAPT
SCHEMBL10165579 0.80 MEN1 (0.62) MEN1KMT2AHTTPOLBMAPT
SCHEMBL10165447 0.80 MEN1 (0.62) MEN1KMT2AHTTPOLBMAPT
SCHEMBL10165501 0.80 MEN1 (0.62) MEN1KMT2AHTTPOLBMAPT
SCHEMBL28921743 0.80 MEN1 (0.50) MEN1KMT2AHTTPOLBMAPT
SCHEMBL10165449 0.79 MEN1 (0.65) MEN1KMT2APOLBMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3565 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
WO-2025094125-A1 AN AGROCHEMICAL COMBINATION UPL MAURITIUS LIMITED (MU) 2025-05-08 WO claimed
US-20230082089-A1 A SYNERGISTIC AGROCHEMICAL COMBINATION UPL LIMITED (IN) 2023-03-16 US claimed
EP-4125382-A1 HERBICIDAL COMBINATION UPL Corporation Limited (MU) 2023-02-08 EP claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
EP-3247698-B1 CRYSTALLINE MODIFICATION OF PROPANIL UPL LTD (IN) 2022-10-19 EP claimed
EP-4046490-A1 AN IMPROVED HERBICIDAL FORMULATION UPL Limited (IN) 2022-08-24 EP claimed
US-8288318-B2 2-(poly-substituted aryl)-6-amino-5-halo-4-pyrimidinecarboxylic acids and their use as herbicides DOW AGROSCIENCES, LLC. (US) 2012-10-16 US claimed
US-20120195974-A1 CONTROLLING MEALYBUGS DOW AGROSCIENCES LLC (US) 2012-08-02 US claimed
WO-2012103393-A2 CONTROLLING MEALYBUGS DOW AGROSCIENCES LLC (US) 2012-08-02 WO claimed
WO-2012061290-A2 PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO DOW AGROSCIENCES LLC (US) 2012-05-10 WO claimed
WO-2012061288-A1 PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO DOW AGROSCIENCES LLC (US) 2012-05-10 WO claimed
US-20120110701-A1 PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO DOW AGROSCIENCES LLC (US) 2012-05-03 US claimed
US-20120110702-A1 Pesticidal Compositions and Processes Related Thereto CORTEVA AGRISCIENCE LLC 2012-05-03 US claimed
US-20110190133-A1 2-(POLY-SUBSTITUTED ARYL)-6-AMINO-5-HALO-4-PYRIMIDINECARBOXYLIC ACIDS AND THEIR USE AS HERBICIDES DOW AGROSCIENCES LLC 2011-08-04 US claimed
WO-2010022251-A2 GABA/PESTICIDAL COMBINATIONS PLANT HEALTH CARE, INC. (US) 2010-02-25 WO claimed
US-20100048397-A1 GABA/Pesticidal Combinations PLANT HEALTH CARE, INC. 2010-02-25 US claimed