SCHEMBL13458583

SCHEMBL13458583

CC(C)=NC(=O)c1csc(CN2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.46
ACKR3 P25106 4/20 0.44
VEGFA P15692 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
PIK3CD O00329 3/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
MAP4K4 O95819 1/20 0.37
BAZ2A Q9UIF9 1/20 0.37
GBA1 P04062 1/20 0.37
TLR8 Q9NR97 1/20 0.36
GLS O94925 1/20 0.35
FGFR1 P11362 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL348893 0.86 HRH3 (0.46) HRH3ACKR3VEGFAEGLN1PIK3CD
SCHEMBL3265007 0.85 ACKR3 (0.49) HRH3ACKR3VEGFAEGLN1PIK3CD
SCHEMBL348818 0.82 ACKR3 (0.51) HRH3ACKR3VEGFAEGLN1PIK3CD
SCHEMBL347902 0.82 HRH3 (0.44) HRH3ACKR3PIK3CD
SCHEMBL6183439 0.73 ACKR3 (0.45) ACKR3VEGFAEGLN1GBA1
SCHEMBL2733360 0.72 CYP3A4 (0.60)
SCHEMBL1929314 0.72 CNR2 (0.51) ACKR3VEGFAEGLN1PIK3CDBAZ2A
SCHEMBL28746914 0.72 ACKR3 (0.47) ACKR3VEGFAEGLN1CHRM2CHRM4
SCHEMBL21579067 0.71 ACKR3 (0.49) ACKR3VEGFAEGLN1PIK3CDCHRM2
SCHEMBL2734028 0.71 ALDH1A1 (0.60) ACKR3VEGFAEGLN1PIK3CDCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025179-A1 1-(4-UREIDOBENZOYL)PIPERAZINE DERIVATIVES N.V. ORGANON (NL) 2010-03-04 WO disclosed