SCHEMBL13458752

SCHEMBL13458752

FC(F)(F)c1ccc(-c2cc(-c3ccc(-c4ccccc4)cc3)c3ccc4c(-c5ccc(-c6ccccc6)cc5)cc(-c5ccc(C(F)(F)F)cc5)nc4c3n2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 5/20 0.59
KIF11 P52732 1/20 0.55
LTB4R Q15722 2/20 0.44
METAP2 P50579 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSPO P30536 1/20 0.43
P2RY14 Q15391 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
ACP1 P24666 1/20 0.43
BACE1 P56817 1/20 0.43
MAOB P27338 1/20 0.43
DGAT1 O75907 1/20 0.43
KCNH2 Q12809 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5931070 0.98 TOP1 (0.60) TOP1KIF11LTB4RMETAP2CYP2C9
SCHEMBL13458749 0.90 TOP1 (0.48) TOP1KIF11METAP2DGAT1KCNH2
SCHEMBL3358457 0.87 ACACA (0.50) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL17899330 0.87 ACACA (0.50) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL1745982 0.87 ACACA (0.50) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL3698074 0.87 ACACA (0.50) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL3358750 0.87 ACACA (0.50) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL14553726 0.85 TOP1 (0.50) TOP1KIF11CYP2C9TSPOP2RY14
SCHEMBL12112655 0.85 ACACA (0.51) TOP1MAPTKDM4ESMN1; SMN2ACACA
SCHEMBL5931163 0.85 TOP1 (0.49) TOP1METAP2MAOBKCNH2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161272-A1 Phenanthrolines BASF SE (DE) 2010-03-10 EP disclosed