SCHEMBL13475426

SCHEMBL13475426

Cc1cccc(N2CCN(CCCn3cccc(O)c3=O)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.61
DRD2 P14416 2/20 0.51
DRD4 P21917 1/20 0.51
DRD3 P35462 1/20 0.51
HTR7 P34969 1/20 0.47
HTR2A P28223 1/20 0.47
HRH1 P35367 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13493143 0.84 HTR7 (0.50) DRD2DRD3HTR7HTR2A
SCHEMBL13496856 0.84 HTR7 (0.50) DRD2DRD3HTR7HTR2A
SCHEMBL8057138 0.84 DRD3 (0.58) DRD2DRD3HTR7HTR2A
SCHEMBL4519876 0.77 KCNH2 (1.00) KCNH2HTR7
SCHEMBL11161100 0.76 KCNH2 (0.80) KCNH2DRD2DRD3HTR7HTR2A
SCHEMBL13711972 0.75 KCNH2 (0.84) KCNH2DRD2HTR7HRH1
SCHEMBL3198969 0.74 KCNH2 (0.72) KCNH2DRD2DRD4DRD3HTR7
SCHEMBL15118465 0.74 EGLN1 (0.50) DRD2HTR2A
SCHEMBL13475441 0.74 KDM1A (0.45) HRH1
SCHEMBL11353566 0.73 KCNH2 (0.80) KCNH2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2151777-A1 Method for screening of 5HT7 receptor ligands based on a new pharmacophore model and a descriptor's profile filter Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-02-10 EP disclosed