SCHEMBL13475701

SCHEMBL13475701

C=C1N(Cc2ccc(Oc3ccccc3)cc2)C(=N)NC1(C)CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 9/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.33
LTA4H P09960 1/20 0.33
PTPRF P10586 1/20 0.32
PTPN2 P17706 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPRB P23467 1/20 0.32
ACP1 P24666 1/20 0.32
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7513751 0.89 LMNA (0.41) CCR5MEN1KMT2ACYP3A4PTPRF
SCHEMBL7516939 0.79 LMNA (0.43) MEN1KMT2AFAAH
SCHEMBL7513640 0.79 MAPK14 (0.52) MEN1KMT2ACYP3A4
SCHEMBL14104839 0.77 ELANE (0.49) MEN1KMT2ACYP3A4
SCHEMBL7532103 0.73 CMA1 (0.45) MEN1KMT2A
SCHEMBL7513704 0.73 MAPK14 (0.47) CYP3A4
SCHEMBL7511268 0.72 SMN1; SMN2 (0.41) KMT2A
SCHEMBL7516805 0.71 BACE1 (0.47) MEN1KMT2APTPN1
SCHEMBL8290131 0.71 SMN1; SMN2 (0.41) MEN1KMT2ACYP3A4
SCHEMBL7534170 0.70 BACE1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2153832-A2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-02-17 EP disclosed