SCHEMBL13480558

SCHEMBL13480558

CCOC(=O)Nc1nc2ccc(C)cc2s1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.77
RAB9A P51151 12/20 0.71
NPC1 O15118 11/20 0.71
SMN1; SMN2 Q16637 8/20 0.71
ALDH1A1 P00352 4/20 0.71
TP53 P04637 3/20 0.71
L3MBTL1 Q9Y468 1/20 0.71
DYRK1A Q13627 1/20 0.68
ACP1 P24666 1/20 0.63
KDM4E B2RXH2 4/20 0.61
MAPT P10636 2/20 0.61
STAT1 P42224 1/20 0.60
MITF O75030 1/20 0.60
POLB P06746 1/20 0.60
APEX1 P27695 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
TSHR P16473 1/20 0.60
CLK1 P49759 1/20 0.59
MEN1 O00255 2/20 0.57
NFKB1 P19838 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14113317 0.87 DYRK1A (0.74) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL22208435 0.87 RAB9A (0.76) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL14189674 0.85 PTPN1 (0.61) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8689148 0.83 NPC1 (1.00) RAB9ANPC1SMN1; SMN2ALDH1A1TP53
SCHEMBL14189669 0.83 RAB9A (0.74) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL11161571 0.83 KMT2A (0.73) RAB9ANPC1SMN1; SMN2ALDH1A1DYRK1A
SCHEMBL7662743 0.83 RAB9A (0.63) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL17090573 0.83 LCK (0.69) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL29506738 0.83 LCK (0.69) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL14189676 0.82 CLK1 (0.58) PTPN1RAB9ANPC1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7659404-B2 Broad spectrum 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors TIBOTEC PHARMACEUTICALS LTD. (IE) 2010-02-09 US disclosed