SCHEMBL1348720

SCHEMBL1348720

NCCNS(=O)(=O)c1ccc(C#Cc2cnn3c(C(F)(F)F)cc(-c4cccc(C(F)(F)F)c4)nc23)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KDM4E B2RXH2 7/20 0.38
ALDH1A1 P00352 5/20 0.38
CYP3A4 P08684 2/20 0.38
GAA P10253 2/20 0.38
HSD17B10 Q99714 4/20 0.38
MAPK1 P28482 2/20 0.38
P2RY14 Q15391 3/20 0.37
ITGB3 P05106 6/20 0.37
ITGA2B P08514 6/20 0.37
CYP1A2 P05177 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1348077 0.92 P2RY14 (0.43) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1347974 0.90 KDM4E (0.38) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1348706 0.87 HPGD (0.44) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1348841 0.87 HPGD (0.44) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1346622 0.85 HPGD (0.39) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL2825050 0.85 HPGD (0.44) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1348463 0.82 KDM4E (0.37) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1348776 0.82 LMNA (0.36) KDM4EALDH1A1MAPTTHRB
SCHEMBL1348340 0.81 HPGD (0.40) HPGDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL1348251 0.81 CDK2 (0.39) HPGDCYP2C9CYP2C19KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4801724-B2 2011-10-26 JP claimed
US-8063048-B2 Acetylenyl-pyrazolo-pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-11-22 US disclosed