SCHEMBL13495653

SCHEMBL13495653

Cc1nc2ccccc2n1-c1ccc(-n2c(C)nc3ccc(F)cc32)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.66
HTT P42858 1/20 0.66
GRIA1 P42261 1/20 0.51
CACNG8 Q8WXS5 1/20 0.51
CACNG2 Q9Y698 1/20 0.51
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.49
PIK3CD O00329 2/20 0.48
PIK3CA P42336 2/20 0.48
MTOR P42345 2/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GLA P06280 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ALDH3A1 P30838 1/20 0.46
GSR P00390 1/20 0.45
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3052790 0.91 MAPK1 (0.65) MAPK1HTTALDH1A1PIK3CDPIK3CA
SCHEMBL22507416 0.91 MAPK1 (0.74) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL13495703 0.88 MAPK1 (0.54) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL13495650 0.87 HTT (0.50) MAPK1HTTPIK3CDPIK3CAMTOR
SCHEMBL13495748 0.85 PIK3CA (0.54) MAPK1HTTALDH1A1PIK3CDPIK3CA
SCHEMBL22507417 0.83 MAPK1 (0.68) MAPK1HTTTSHRALDH1A1KDM4E
SCHEMBL22507480 0.83 HTT (0.67) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL13495698 0.82 PIK3CA (0.53) MAPK1HTTPIK3CDPIK3CAMTOR
SCHEMBL13495701 0.81 APP (0.50) ALDH1A1KDM4ESMN1; SMN2L3MBTL1GLA
SCHEMBL13495695 0.81 NPC1 (0.58) MAPK1HTTALDH1A1PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012745-A2 BENZIMIDAZOLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-02-04 WO disclosed