SCHEMBL13504665

SCHEMBL13504665

CC(C)(C)OC(=O)Nc1cc(-c2cc(F)ccc2-c2ccn(-c3ccc4nnc(N)n4n3)n2)ccn1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.37
RIPK3 Q9Y572 1/20 0.37
CDK9 P50750 2/20 0.34
AAK1 Q2M2I8 4/20 0.34
NTRK1 P04629 4/20 0.34
TGFBR1 P36897 1/20 0.33
NR3C2 P08235 2/20 0.33
KMT2A Q03164 2/20 0.33
PIK3C3 Q8NEB9 1/20 0.33
MEN1 O00255 1/20 0.33
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
CDK3 Q00526 1/20 0.32
CDK5 Q00535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5350862 0.84 IRAK4 (0.39) IRAK4RIPK3CDK9NR3C2GSK3B
SCHEMBL5353510 0.75 MAPK10 (0.39) IRAK4RIPK3TGFBR1NR3C2
SCHEMBL5352686 0.75 KCNH2 (0.38) IRAK4RIPK3CDK9NR3C2
SCHEMBL5347459 0.74 MAPK14 (0.40) IRAK4RIPK3
SCHEMBL1104982 0.71 RIPK3 (0.44) IRAK4RIPK3CDK9AAK1TGFBR1
SCHEMBL5350912 0.69 NR3C2 (0.39) IRAK4RIPK3CDK9NR3C2
SCHEMBL5350212 0.68 CDK9 (0.40) IRAK4CDK9TGFBR1
SCHEMBL5352200 0.67 IRAK4 (0.42) IRAK4RIPK3CDK9NR3C2PIK3C3
SCHEMBL15885857 0.67 IRAK4 (0.55) IRAK4AAK1TGFBR1PIK3C3GSK3B
SCHEMBL29402022 0.66 ATR (0.46) IRAK4RIPK3CDK9TGFBR1PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553096-B1 PYRAZOLE COMPOUNDS UBE INDUSTRIES (JP) 2012-10-31 EP disclosed