SCHEMBL13521950

SCHEMBL13521950

CC(C)(C)C(=O)Nc1ccc(Oc2cc(CC(=O)O)cc(C(F)(F)F)c2)c(CS)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
RXRA P19793 4/20 0.39
RXRB P28702 4/20 0.39
RXRG P48443 4/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
THRB P10828 2/20 0.37
THRA P10827 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
P2RX4 Q99571 1/20 0.35
FFAR1 O14842 1/20 0.35
NR3C1 P04150 1/20 0.35
NR1H4 Q96RI1 2/20 0.35
S1PR1 P21453 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13521902 0.89 CYP3A4 (0.39) CYP3A4LMNAPOLBSLC6A2SLC6A4
SCHEMBL349585 0.86 CYP3A4 (0.52) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL348413 0.86 CYP3A4 (0.52) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL13521968 0.86 CYP3A4 (0.51) CYP3A4PTGDR2SLC6A3P2RX4CYP2C9
SCHEMBL12375407 0.86 CYP3A4 (0.45) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL349569 0.85 CYP3A4 (0.45) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL27807724 0.81 CYP3A4 (0.43) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL349570 0.80 PTGDR2 (0.40) CYP3A4RXRARXRBRXRGPTGDR2
SCHEMBL16510020 0.79 CYP3A4 (0.47) CYP3A4RXRARXRBRXRGLMNA
SCHEMBL13521934 0.78 CYP3A4 (0.62) CYP3A4PTGDR2LMNANR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010003127-A2 ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-01-07 WO disclosed