SCHEMBL13539628

SCHEMBL13539628

COc1c(C)ncc(CN2CC(=O)c3c(Cl)nc(N)nc32)c1C

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 19/20 0.55
HSP90AA1 P07900 19/20 0.54
HSP90B1 P14625 1/20 0.38
TRAP1 Q12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13539741 0.89 HSP90AB1 (0.47) HSP90AB1HSP90AA1
SCHEMBL13616277 0.83 HSP90AB1 (0.70) HSP90AB1HSP90AA1
SCHEMBL13539735 0.81 HSP90AA1 (0.48) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL13539714 0.81 HSP90AA1 (0.71) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL13539719 0.80 HSP90AA1 (0.46) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL13539631 0.79 HSP90AA1 (0.47) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL14567691 0.78 HSP90AA1 (0.46) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL13539447 0.78 HSP90AA1 (0.54) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL13539630 0.78 HSP90AA1 (0.51) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL14567690 0.77 HSP90AA1 (0.41) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2145888-A1 Deazapurine derivatives as HSP90-Inhibitors Conforma Therapeutics Corporation (US) 2010-01-20 EP disclosed