SCHEMBL13539655

SCHEMBL13539655

CBc1c(C)cnc(CN2C(=O)Cc3c(Cl)nc(N)nc32)c1C

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 16/20 0.50
TRAP1 Q12931 9/20 0.50
HSP90B1 P14625 7/20 0.50
HSP90AB1 P08238 11/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391833 0.87 HSP90AA1 (0.57) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL13539742 0.85 HSP90AA1 (0.59) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL1052242 0.83 HSP90AA1 (0.62) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL5566304 0.82 HSP90AA1 (0.53) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL12615628 0.81 HSP90AA1 (0.59) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL1060933 0.77 HSP90AA1 (0.56) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL12651963 0.74 HSP90AA1 (0.59) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL1060436 0.74 TRAP1 (0.66) HSP90AA1TRAP1HSP90B1
SCHEMBL1079346 0.70 HSP90AA1 (0.60) HSP90AA1TRAP1HSP90B1HSP90AB1
SCHEMBL1078262 0.70 HSP90AA1 (0.57) HSP90AA1TRAP1HSP90B1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2145888-A1 Deazapurine derivatives as HSP90-Inhibitors Conforma Therapeutics Corporation (US) 2010-01-20 EP disclosed